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Deprecated: Implicit conversion from float 215.6 to int loses precision in C:\Inetpub\vhosts\kidney.de\httpdocs\pget.php on line 534 Oncotarget 2017 ; 8 (12): 20452-61 Nephropedia Template TP
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Homeodomain-interacting protein kinase 2 (HIPK2): a promising target for anti-cancer therapies #MMPMID28107201
Feng Y; Zhou L; Sun X; Li Q
Oncotarget 2017[Mar]; 8 (12): 20452-61 PMID28107201show ga
The HIPK2 (serine/threonine homeodomain-interacting protein kinase 2) is a ?caretaker? gene, its inactivation increases tumorigenicity while its activation inhibits tumor growth. This report reviews the anti-tumorigenic mechanisms of HIPK2, which include promotion of apoptosis, inhibition of angiogenesis in hypoxia, prevention of tumor invasion/metastasis and attenuation of multidrug resistance in cancer. Additionally, we summarize conditions or factors that may increase HIPK2 activity.